Clinical Stage Programs
Program
                                    MOA
                                    Indications
                                    IND
                                    Phase I
                                    Phase II
                                    Phase III
                                    Rights
                                LM-302
                                            Anti-Claudin18.2 ADC
                                            3L+ GC/GEJ
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-302
                                            Anti-Claudin18.2 ADC
                                            1L GC/GEJ
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-302
                                            Anti-Claudin18.2 ADC
                                            PDAC
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-108
                                            Anti-CCR8 mAb
                                            MSI-H tumors
                                             
                                                                     
                                                                    
                                                ex-China available                                                                                                
                                            
                                        LM-108
                                            Anti-CCR8 mAb
                                            2L GC/GEJ
                                             
                                                                     
                                                                    
                                                ex-China available                                                                                                
                                            
                                        LM-101
                                            Anti-SIRPα mAb
                                            Solid tumors & hematologic malignancies
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-305
                                            Anti-GPRC5D ADC
                                            Multiple Myeloma
                                             
                                                                     
                                                                    
                                                AstraZeneca (Global)                                                                                                
                                            
                                        LM-24C5
                                            CEACAM5 BsAb
                                            CRC, GI cancer, lung cancer
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-299
                                            anti-PD-1 x anti-VEGF BsAb
                                            Solid tumors
                                             
                                                                     
                                                                    
                                                MSD (Global)                                                                                                
                                            
                                        LM-168
                                            Anti-CTLA4 (TME specific)
                                            Solid tumors
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-2417
                                            Anti-NaPi2b BsAb
                                            Lung cancer, ovarian cancer
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        
                                    Clinical Stage Programs                                
                                
                                                    LM-302                                                
                                                
                                                    3L+ GC/GEJ                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Anti-Claudin18.2 ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-302                                                
                                                
                                                    1L GC/GEJ                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Anti-Claudin18.2 ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-302                                                
                                                
                                                    PDAC                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Anti-Claudin18.2 ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-108                                                
                                                
                                                    MSI-H tumors                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Anti-CCR8 mAb                                                
                                                
                                                    Rights
                                                
                                                
                                                    ex-China available                                                                                                        
                                            
                                                    LM-108                                                
                                                
                                                    2L GC/GEJ                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Anti-CCR8 mAb                                                
                                                
                                                    Rights
                                                
                                                
                                                    ex-China available                                                                                                        
                                            
                                                    LM-101                                                
                                                
                                                    Solid tumors & hematologic malignancies                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Anti-SIRPα mAb                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-305                                                
                                                
                                                    Multiple Myeloma                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Anti-GPRC5D ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    AstraZeneca (Global)                                                                                                        
                                            
                                                    LM-24C5                                                
                                                
                                                    CRC, GI cancer, lung cancer                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    CEACAM5 BsAb                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-299                                                
                                                
                                                    Solid tumors                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    anti-PD-1 x anti-VEGF BsAb                                                
                                                
                                                    Rights
                                                
                                                
                                                    MSD (Global)                                                                                                        
                                            
                                                    LM-168                                                
                                                
                                                    Solid tumors                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Anti-CTLA4 (TME specific)                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-2417                                                
                                                
                                                    Lung cancer, ovarian cancer                                                
                                            IND
                                                Phase I
                                                Phase II
                                                Phase III
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Anti-NaPi2b BsAb                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            Preclinical Stage Programs
Program
                                    MOA
                                    Indications
                                    Discovery
                                    PCC
                                    IND-enabling
                                    Rights
                                LM-350
                                            anti-CDH17 ADC
                                            CRC, PDAC, GC
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-364
                                            Undisclosed ADC
                                            NSCLC, HNSCC, UC
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-338
                                            Undisclosed ADC
                                            CRC, NSCLC, GC
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-359
                                            Undisclosed ADC
                                            HCC
                                             
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-319
                                            Undisclosed ADC
                                            TNBC, lung cancer
                                             
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-316
                                            Undisclosed ADC
                                            NSCLC, OC, TNBC
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-339
                                            Undisclosed ADC
                                            NSCLC, OC
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        LM-2199
                                            Undisclosed BsAb
                                            NSCLC, CRC, HNSCC, GC
                                             
                                                                     
                                                                    
                                                Global available                                                                                                
                                            
                                        
                                    Clinical Stage Programs                                
                                
                                                    LM-350                                                
                                                
                                                    CRC, PDAC, GC 
                                                
                                            Discovery
                                                PCC
                                                IND-enabling
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    anti-CDH17 ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-364                                                
                                                
                                                    NSCLC, HNSCC, UC 
                                                
                                            Discovery
                                                PCC
                                                IND-enabling
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Undisclosed ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-338                                                
                                                
                                                    CRC, NSCLC, GC 
                                                
                                            Discovery
                                                PCC
                                                IND-enabling
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Undisclosed ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-359                                                
                                                
                                                    HCC 
                                                
                                            Discovery
                                                PCC
                                                IND-enabling
                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Undisclosed ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-319                                                
                                                
                                                    TNBC, lung cancer 
                                                
                                            Discovery
                                                PCC
                                                IND-enabling
                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Undisclosed ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-316                                                
                                                
                                                    NSCLC, OC, TNBC 
                                                
                                            Discovery
                                                PCC
                                                IND-enabling
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Undisclosed ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-339                                                
                                                
                                                    NSCLC, OC 
                                                
                                            Discovery
                                                PCC
                                                IND-enabling
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Undisclosed ADC                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                            
                                                    LM-2199                                                
                                                
                                                    NSCLC, CRC, HNSCC, GC 
                                                
                                            Discovery
                                                PCC
                                                IND-enabling
                                             
                                                             
                                                            
                                                    MOA
                                                
                                                
                                                    Undisclosed BsAb                                                
                                                
                                                    Rights
                                                
                                                
                                                    Global available                                                                                                        
                                             
                     
         
    